RANKING of DRUGS fitting to SARS proteinase model既存医薬品データのうち、SARSプロテアーゼのリガンドとして適すると推定されるものを調査し、ランキング付けいたしました。
RANK DRUG name 1 fradiomycin_sulfate 2 tobramycin 3 kanamycin_sulfate 4 netilmicin_sulfate 5 cefmenoxime_hydrochloride 6 ioversol 7 ribostamycin_sulfate 8 cefpiramide_sodium 9 micronomicin_sulfate 10 nelfinavir 11 ribavirin_3phosphate 12 cefotetan 13 aztreonam 14 latamoxef_sodium 15 mitoxantrone_hydrochloride 16 ioxilan 17 deferoxamine_mesilate 18 amikacin_sulfate 19 aspoxicillin 20 sennoside 21 salazosulfapyridine 22 argatroban 23 bergenin 24 iomeprol 25 famotidine 26 bekanamycin_sulfate 27 cabergoline 28 carumonam_sodium 29 cefteram_pivoxil 30 cefotetan_sodium 31 riboflavin_sodium_phosphate 32 cefotiam_hydrochloride 33 iohexol 34 amogastrin 35 oxiglutatione 36 lincomycin_hydrochloride 37 doxorubicin_hydrochloride 38 cefminox_sodium 39 hexoprenaline_sulfate 40 ritonavir 41 cocarboxylase 42 glucosulfone_sodium 43 streptomycin_sulfate 44 sisomicin_sulfate 45 astromicin_sulfate 46 dibekacin_sulfate 47 folic_acid 48 tetracycline 49 ceftezole_sodium 50 clindamycin_phosphate The nelfinavir structure of rank 10 complexed with SARS proteinase was shown in the figure of O.